Wednesday, 31 May 2006: 8:30 AM-12:00 PM
Regency Ballroom A (Hyatt Regency Milwaukee)
Medicinal Chemistry (MEDI)
New Strategies for Modern Medicinal Chemistry I
Invited presentations in Medicinal Chemistry. Topics will include pharmaceutical drug discovery towards antiviral agents, cancer therapy, and neurological disorders.
Organizer:Keith McDaniel
Presider:Keith McDaniel
8:30 AMIntroductory Remarks
8:35 AMRational Drug Design. Where it has been and where might it go in the 21st Century
Daniel H. Rich
9:20 AMThe search for the next generation of HIV protease inhibitors
David A. DeGoey
10:05 AMBreak
10:30 AMThe design of hepatitis C protease inhibitors and the discovery of VX-950
Robert B. Perni
11:15 AMWhat molecular forces could possibly be involved in stabilizing the topoisomerase I-DNA-inhibitor ternary cleavage complex and what do the answers tell us about how to design more effective topoisomerase I inhibitors?
Mark Cushman, Xiangshu Xiao, Alexandra Ioanoviciu, Andrew Morrell, Muthukaman Nagarajan, Yves Pommier, Smitha Antony, Glenda Kohlhagen, Christophe Marchand, Kurt W. Kohn, Bart L. Staker, Alex B. Burgin, Lance Stewart

Back to The 37th Great Lakes Regional Meeting (May 31- June 2, 2006)