Monday, 23 May 2005: 1:00 PM-4:00 PM | |||
Room 203 (Science & Engineering Resource Center) | |||
Medicinal Chemistry (MEDI) | |||
GPCR / Virtual Screening | |||
| This session is intended to cover 4 or 5 30 minute presentations giving an overview of current drug discovery efforts which target G protein-coupled receptors for therapeutic indications. | |||
| Organizer: | Robert Goodnow | ||
| Workshop Leader: | Dr. Shawn Erickson | ||
| 1:00 PM | Introductory Remarks Shawn Erickson | ||
| 1:05 PM | 224 | Ligand Twisting and Counterion Switching in Rhodopsin Activation Thomas P. Sakmar | |
| 1:35 PM | 225 | Using Designed Peptide Panels for De-risking GPCR Projects Waleed Danho | |
| 2:05 PM | 226 | GPCR Ligands from Enzyme Targeted Libraries Michael Ohlmeyer | |
| 2:35 PM | Coffee Break | ||
| 3:00 PM | 227 | Discovery and Development of the First Centrally Active mGluR5 Positive Allosteric Modulators Craig Lindsley | |
| 3:30 PM | 228 | A LMW CCR5 Antagonist in Combination with CsA Prolongs Graft Survival in Life Supporting Kidney TX Model in Cynomolgus Monkeys Gerhard Thoma | |
Back to The 37th Middle Atlantic Regional Meeting (May 22-25, 2005)