Monday, 5 June 2006: 1:25 PM-5:30 PM
Cocoa 6 (Hershey Lodge and Convention Center)
Organic and Medicinal Chemistry (ORGM)
Benchtop-to-Pilot Plant
Designing and implementing a safe and robust process requires a combination of synthetic creativity, development and utilization of new technologies, and effective engineering. Speakers in this session will address recent challenges in pharmaceutical process chemistry and their strategies for a successful, scalable process.
Sponsor: Pfizer
Organizer:Jennifer Rutherford
Presider:Jennifer Rutherford
1:25 PMIntroductory Remarks
1:30 PMTailored solutions for the formation of amide bonds in large scale
Silvina García Rubio
2:05 PMApplication of flow microreactor technology in process research
Xini Zhang
2:40 PMDevelopment of a Practical Synthesis of a GABAa á 2,3-Selective Allosteric Modulator
R. Scott Hoerrner, Mark S. Jensen, Wenjie Li, Dorian P. Nelson, Gary J. Javadi, Peter G. Dormer, Dongwei Cai, Robert D. Larsen
3:15 PMBreak
3:25 PMAEW541: A Challenge to Process Chemists
Joel S. Slade, Joginder Bajwa, Kapa Prasad, Hui Liu, John Calienni, James Vivelo, David Parker, Guang-Pei Chen, Edwin Villhauer
4:00 PMIntegration of Lithiation and Coupling Reactions into a Continuous Process as an Alternative to a Cryogenic Batch Synthesis
Chenchi Wang, Prashant Deshpande, Wendy Yang, Thomas LaPorte
4:35 PMProcess development and large-scale synthesis of a PDE-IV inhibitor
Brenda Pipik, David A. Conlon, Antoinette Drahus-Paone, Guo-Jie Ho, Roy Helmy, Yao-Jun Shi, James M. McNamara, J. Michael Williams
5:10 PMAir-stable Palladium-Phosphine based catalysts for challenging Carbonylation and Coupling reactions
Thomas Colacot

Back to The 38th Middle Atlantic Regional Meeting (June 4-7, 2006)