Tuesday, 6 June 2006: 1:30 PM-5:00 PM
Magnolia C-D (Hershey Lodge and Convention Center)
Organic and Medicinal Chemistry (ORGM)
MARM Honors: The Alfred Burger Award, Part II
This symposium honors the ACS Division of Medicinal Chemistry Burger Award and consists of three invited speakers who have won this national award, three additional invited speakers, and a select number of contributed papers.
Sponsor: ACS Division of Medicinal Chemistry and Merck and Co
Organizer:Stephen C. Waller
Presider:Alan Cooper
1:30 PMIntroductory Remarks
1:35 PMQuantum mechanics and the molecules of medicinal chemistry
Lou Massa, Lulu Huang, Jerome Karle
2:00 PMDesign and Synthesis of Thrombin Receptor (PAR-1) Antagonists
William Greenlee, Samuel Chackalamannil, Mariappan Chelliah, Martin Clasby, Michael Czarniecki, Keith Eagen, Xiaobang Gao, Dario Doller, Zhiyong Hu, Yan Lin, Hsing-An Tsai, Yuguang Wang, Yan Xia
2:50 PMBreak
3:05 PMSome reflections on the design of GPCR agonists with privileged structures
Arthur A. Patchett
3:55 PMAre heterodimeric G protein-coupled receptors viable targets for medicinals? Opioid receptors as proof of concept
Philip S. Portoghese
4:55 PMConcluding Remarks

Back to The 38th Middle Atlantic Regional Meeting (June 4-7, 2006)