Friday, 3 November 2006: 8:00 AM-12:00 PM
Estes A (Augusta Marriott Hotel and Suites)
Medicinal Chemistry (17)
Chemistry of drug abuse (MEDI, BIOL)
Sponsor: ACS Division of Medicinal Chemistry
Organizer:Bruce Blough
Presider:Bruce Blough
8:00 AMIntroductory Remarks
8:10 AMA novel series of kappa opioid antagonists based on JDTic: Identifying structural features that modulate potency, selectivity and function
Scott P. Runyon, Hernan Navarro, James Thomas, F. Ivy Carroll
8:40 AMSynthesis of phenylmorphan-based antagonists of the kappa opioid receptor
James B. Thomas, Matt S. Melvin, Michel C. Nuckols, Hernan A. Navarro, F. Ivy Carroll
9:10 AMRecent advances in neurotransmitter releasers
Bruce E. Blough, Kevin Page, Tony Landavazo, John Partilla, Richard Rothman
9:40 AMBreak
10:00 AMSAR of the salvinorin A scaffold: discovery of selective mu opioids
Thomas E. Prisinzano
10:30 AMDevelopment of ligands for nicotinic acetylcholine receptors (nAChRs) as potential pharmacotherapies for treating smokers
F. Ivy Carroll, Hernán A. Navarro, Bruce E. Blough, Billy R. Martin, M. Imad Damaj, Ronald J. Lukas, Charles W. Luetje

Back to The 58th Southeast Regional Meeting (November 1-4, 2006)