Saturday, October 27, 2007: 8:40 AM-12:00 PM
Redbud C (Greenville Hyatt Regency Hotel)
Medicinal and Biochemistry (3)
General Medicinal Chemistry
General medicinal chemistry posters and oral presentations.
Presider:Dev P. Arya
Organizer:William T. Pennington
8:40 AMComparative Carcinogenicity of Oxidized Metabolites of Preprocarcinogens and Procarcinogens with Aromatic Structural Types ArX and ArCH2X
James W. Flesher, Jamie Horn, Andreas F. Lehner
9:00 AMAntibody-Catalyzed Oxidation of &Delta9-Tetrahydrocannabinol &Delta9-THC
Andrew P. Brogan, Lisa M. Eubanks, George F. Koob, Tobin J. Dickerson, Kim D. Janda
9:20 AMAntiproliferative Bistramides of the Marine Ascidian Trididemnum Sp. from Madagascar
Brian T. Murphy, Shugeng Cao, Peggie Brodie, David G. I. Kingston, Jean Maharavo
9:40 AMBreak
10:00 AMSynthesis and Evaluation of Lysophosphatidylcholine Analogs as Tools to Determine Crucial Autotaxin Substrate Characteristics
E. Jeffrey North, Daniel L. Baker, Abby L. Parrill
10:20 AMDNA Conformational Changes Induced by a Highly Charged, Cytotoxic Platinum-Based Bisintercalator
Jayati Roy Choudhury, Rajsekhar Guddneppanavar, Gregory L. Kucera, Gilda Saluta, Ulrich Bierbach
10:40 AMDesign Synthesis and Biological Evaluation of Biomimmetic Analogues of Colchicine: α-2,3,4-Trimethoxyphenyl-β-Acetamido Naphthalene
Anthony J. Fowler, Craig Ogle, James P. Snyder, Ana Alcaraz
11:00 AMSynthesis of Novel Selective Inhibitors of Human Intestinal Carboxylesterase Designed to Ameliorate the Delayed Diarrhea Associated with CPT-11 Treatment
Latorya D. Hicks, Janice L. Hyatt, Lyudmila Tsurkan, Jason Hatfield, Carol Edwards, Philip M. Potter, Randy M. Wadkins
11:20 AMSynthesis of Novel GABA Analogs and Their Activity at GABAC Receptors
Robert F. Standaert, Jun Yan, Niraj J. Muni, David R. Pepperberg

Back to The Southeastern Regional Meeting (October 24 – 27, 2007)