Bioorganic Chemistry Session II [Oral]

Friday, 23 October 2009: 08:30-16:50
103-B (Puerto Rico Convention Center)
Presiders:
Cornelis Vlaar and Eliud Hernandez, Ph.D.
Organizer:
Néstor M. Carballeira, Ph.D.
8:30 AM
Introductory Remarks
8:35 AM
471
Four Proline-Containing Cycloheptapeptides From the Caribbean Marine Sponge Prosuberites Laughlini
Brunilda Vera, University of Puerto Rico, Rio Piedras Campus; Jan Vicente, University of Puerto Rico; Abimael D. Rodríguez, University of Puerto Rico, Rio Piedras Campus
8:55 AM
472
Total Synthesis and Biological Evaluation of 8 Epi-Lucentamycin A
R. Nathan Daniels, Vanderbilt University; Craig W. Lindsley, Vanderbilt University
9:15 AM
473
Solid-Phase Phosphitylating Reagents: Design and Application in the Synthesis of Phosphorylated Biomolecules
Yousef Ahmadi Beni, Assistant Professor of Chemistry, Columbus State University; Keykavous Parang, University of Rhode Island
9:35 AM
474
Corallolides A and B: A Novel Class of Diterpenes Isolated From the Caribbean Gorgonian Coral Pseudopterogorgia Bipinnata
Claudia A. Ospina, Ph.D., University of Puerto Rico at Cayey; Abimael D. Rodríguez, Ph.D., University of Puerto Rico, Rio Piedras Campus
9:55 AM
Break
10:15 AM
475
Antibiotic Cytosporone E: Analog Synthesis Via Selective Deletion of Oxygen Atoms and the Incorporation of Nitrogen
Thomas L. Jenkins, College of Charleston; Justin K. Wyatt, College of Charleston
10:35 AM
476
Tetrahydro-4-Quinolinamines Identified as Novel P2Y1 Receptor Antagonists
Angel I. Morales Ramos, Ph.D., University of Puerto Rico - Mayagüez Campus; John Mecom, GlaxoSmithKline; Todd L. Graybill, Ph.D., GlaxoSmithKline; Joseph P. Marino Jr., Ph.D., GlaxoSmithKline
10:55 AM
477
Synthesis of Cyclic 1,2-Disulfides and Cyclic 1,2-Thiosulfinates as Inhibitors of Thioredoxin Reductase
Eory M. Madera- Miranda, University of Puerto Rico, Medical Sciences Campus, School of Pharmacy; Sandraliz Espinosa, University of Puerto Rico, Medical Sciences Campus, School of Pharmacy; Janice Santiago, University of Puerto Rico, Medical Sciences Campus, School of Pharmacy; Marianela Perez-Torrez, University of Puerto Rico, Medical Sciences Campus, School of Pharmacy; Cornelis Vlaar, University of Puerto Rico, Medical Sciences Campus, School of Pharmacy
11:35 AM
479
Synthesis and Anti-Breast Cancer Activity of Novel 1, 3, 4, 8-Tetrahydropyrrolo [4, 3, 2-De]Quinolin-8(1H)-One Alkaloid Analogs
Sadanandan E. Velu, The University of Alabama at Birmingham; Dwayaja H. Nadkarni, The University of Alabama at Birmingham; Srinivasan Murugesan, The University of Alabama at Birmingham
11:55 AM
Lunch Break
1:25 PM
480
Biselisabethoxanes A-D, An Unusual Family of Bisditerpenes From the Gorgonian Coral Pseudopterogorgia Elisabethae
Abimael D. Rodríguez, University of Puerto Rico, Rio Piedras Campus; Ileana I. Rodríguez, University of Puerto Rico, Rio Piedras Campus
1:45 PM
481
SAR Side Chain Derivatives of the Antibiotic Cytosporone E
Erin M. Cartwright, College of Charleston; Justin K. Wyatt, College of Charleston
2:05 PM
482
2:25 PM
483
Functional Reconstitution of the Integral Membrane Enzyme, His-Ste14p, in Synthetic Bolalipid Membrane Vesicles
Wilma Febo-Ayala, University of Puerto Rico-Mayaguez; Shakira L. Morera-Felix, Purdue University; Christine A. Hrycyna, Purdue University; David H. Thompson, Purdue University
2:45 PM
484
Small Molecule Inhibitors of Rac1 as Anti-Invasive Breast Cancer Compounds
Eliud Hernández, School of Pharmacy, Medical Sciences Campus, University of Puerto Rico; Alina De la Mota, School of Medicine, Medical Sciences Campus, University of Puerto Rico; Suranganie Dharmawardhane, School of Medicine, Medical Sciences Campus, University of Puerto Rico; Cornelis P. Vlaar, School of Pharmacy, Medical Sciences Campus, University of Puerto Rico
3:05 PM
Break
3:20 PM
485
Synthesis and Screening of Sigma Receptor Ligands for Post-Stroke Therapy
Michelle Y. Cortes-Salva, University of South Florida; Be-Lan Ngugen, University of South Florida; Adam Behensky, University of South Florida; Keith Pennypacker, University of South Florida; Javier Cuevas, University of South Florida; Jon Antilla, University of South Florida
3:40 PM
486
Synthesis and Biological Activity of Novel Functionalized 4-Aza-2,3-Didehydropodophyllotoxin Derivatives
Ajay Kumar, PhD, University of Puerto Rico Humacao; Antonio E. Alegria, PhD, University of Puerto Rico Humacao; Christian E. Vélez Gerena, Universidad Metropolitana,; Beatriz Zayas, Universidad Metropolitana,
4:00 PM
487
Development of a Simple and Practically Useful Glycosylation Strategy and Its Application to the Concise Synthesis of Carbohydrate Antigens
Pengfei Wang, University of Alabama at Birmingham; Yun Wang, University of Alabama at Birmingham; Xin Zhang, University of Alabama at Birmingham
See more of: Abstract Submission